MRS2395 [CAS 491611-55-3]
Partner: MedChemexpress LLC
CAS No: | 491611-55-3 |
Applications: | Neuroscience-Neuromodulation |
MW: | 439.94 |
Formula: | C20H30ClN5O4 |
SMILES: | CNC1=C2N=CN(CC(COC(C(C)(C)C)=O)COC(C(C)(C)C)=O)C2=NC(Cl)=N1 |
Description: | MRS2395, an dipivaloyl derivative, is a potent P2Y12 receptor antagonist. MRS2395 inhibits ADP-induced platelet activation with a Ki of 3.6 ?M. MRS2395 inhibits cAMP induced by ADP in rat platelets in the presence of PGE1 with an IC50 of 7 �M. MRS2395 enhances platelet dense granule release in response to TRAP-6[1][2]. |
Shipping Conditions: | Ship at ambient |
Usage: | Research Use Only |
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