(Rac)-Tavapadon [CAS 1643462-64-9] (10mM in DMSO)
Partner: MedChemexpress LLC
| CAS No: | 1643462-64-9 |
| Applications: | Neuroscience-Neurodegeneration |
| MW: | 391.34 |
| Formula: | C19H16F3N3O3 |
| SMILES: | O=C1NC(C(C)=C(C2=CC=C(OC3=NC=CC=C3C(F)(F)F)C=C2C)N1C)=O |
| Purity: | 99.87 |
| Description: | (Rac)-Tavapadon ((Rac)-PF-06649751) is a potent and selective noncatechol dopamine D1 receptor agonist. (Rac)-Tavapadon displays potent full agonism in the GS activation assay as well as partial agonism in the ?-arrestin2 recruitment assay (GS-cAMP, EC50=0.8 nM; ?-arrestin2, EC50=68 nM). (Rac)-Tavapadon has antiparkinsonian activity[1]. |
| Shipping Conditions: | Ship on cold packs |
| Usage: | Research Use Only |
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